- 
                                
                                    
                                        
                                        
                                    
                                    
                                        ~3%
                                          
 
 参考文献:
                                    ARRAY BIOPHARMA INC. COOK, Adam HUNT, Kevin, W. DELISLE, Robert Kirk ROMOFF, Todd CLARK, Christopher, T. KIM, Ganghyeok CORRETTE, Christopher, P. DOHERTY, George, A. BURGESS, Laurence, E. Patent: WO/75 A,   Location in patent: Page/Page column 4  WO /75 A
                                 
- 
                                
                                    
                                        
                                        
                                    
                                        
                                        
                                    
                                    
                                        ~95%
                                          
 
 参考文献:
                                    Matsufuji, Tetsuyoshi Shimada, Kousei Kobayashi, Shozo Kawamura, Asuka Fujimoto, Teppei Arita, Tsuyoshi Hara, Takashi Konishi, Masahiro Abe-Ohya, Rie Izumi, Masanori Sogawa, Yoshitaka Nagai, Youko Yoshida, Kazuhiro Takahashi, Hisashi Bioorganic and Medicinal Chemistry Letters, 4 , vol. 4, # 3 p. 75 - 755
                                 
- 
                                
                                    
                                        
                                        
                                    
                                    
                                        ~%
                                          
 
 参考文献:
                                    BAYER INTELLECTUAL PROPERTY GMBH GREUL, Jörg, Nico MANSFIELD, Darren FÜSSLEIN, Martin RIECK, Heiko RIEDRICH, Matthias RODEFELD, Lars KATHER, Kristian MALSAM, Olga LÖSEL, Peter VOERSTE, Arnd SCHWARZ, Hans-Georg ILG, Kerstin GÖRGENS, Ulrich CARLES, Lionel COQUERON, Pierrre-Yves DESBORDES, Philippe MERESSE, Philippe Patent: WO3/6446 A, 3 
                                 
- 
                                
                                    
                                        
                                        
                                    
                                    
                                        ~%
                                          
 
 参考文献:
                                    BAYER INTELLECTUAL PROPERTY GMBH GREUL, Jörg, Nico MANSFIELD, Darren FÜSSLEIN, Martin RIECK, Heiko RIEDRICH, Matthias RODEFELD, Lars KATHER, Kristian MALSAM, Olga LÖSEL, Peter VOERSTE, Arnd SCHWARZ, Hans-Georg ILG, Kerstin GÖRGENS, Ulrich CARLES, Lionel COQUERON, Pierrre-Yves DESBORDES, Philippe MERESSE, Philippe Patent: WO3/6446 A, 3