参考文献:
MERCK SHARP and DOHME CORP. EDMONDSON, Scott, D. CHANG, Lehua KAR, Nam Fung MORRIELLO, Gregori, J. MOYES, Christopher, J. SHEN, Dong-Ming ZHU, Cheng ANTHONY, Neville, J. JONES, Philip SMITH, Graham, F. SCOTT, Mark, E. THOMPSON, Christopher, F. JUNG, Joon CAMMARANO, Carolyn HOFFMAN, Dawn Marie Patent: WO0/5774 A, 0 Location in patent: Page/Page column 49-50 WO 0/05774 A