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MERCK SHARP and DOHME CORP. ElexoPharm GmbH HOYT, Scott, B. PETRILLI, Whitney Lane LONDON, Clare XIONG, Yusheng TAYLOR, Jerry Andrew ALI, Amjad LO, Michael HENDERSON, Timothy, J. HU, Qingzhong HARTMANN, Rolf YIN, Lina HEIM, Ralf BEY, Emmanuel SAXENA, Rohit SAMANTA, Swapan Kumar KULKARNI, Bheemashankar, A. Patent: WO/4888 A, WO /4888 A