~98%
参考文献:
Yeh, Vince S. C. Beno, David W. A. Brodjian, Sevan Brune, Michael E. Cullen, Steven C. Dayton, Brian D. Dhaon, Madhup K. Falls, Hugh D. Gao, Ju Grihalde, Nelson Hajduk, Philip Hansen, T. Matthew Judd, Andrew S. King, Andrew J. Klix, Russel C. Larson, Kelly J. Lau, Yau Y. Marsh, Kennan C. Mittelstadt, Scott W. Plata, Dan Rozema, Michael J. Segreti, Jason A. Stoner, Eric J. Voorbach, Martin J. Wang, Xiaojun Xin, Xili Zhao, Gang Collins, Christine A. Cox, Bryan F. Reilly, Regina M. Kym, Philip R. Souers, Andrew J. Journal of Medicinal Chemistry, 1 , vol. 55, # 4 p. 1751 - 1757