参考文献:
ORTHO-MCNEIL-JANSSEN PHARMACEUTICALS, INC GIJSEN, Henricus, Jacobus, Maria BISCHOFF, Francois Paul ZHUANG, Wei VAN BRANDT, Sven, Franciscus, Anna SURKYN, Michel ZAJA, Mirko BERTHELOT, Didier, Jean-Claude DE CLEYN, Michel, Anna, Jozef MACDONALD, Gregor, James OEHLRICH, Daniel Patent: WO00/94647 A, 00 Location in patent: Page/Page column 64 WO 00/094647 A